• 11 Hits
  • 検索条件 : 絞込み (MeSH = Azepines / pharmacology*)
生物種 リソース名 タイトル
ヒト・動物細胞 StromaNKtert(RCB2350) The BET bromodomain inhibitor CPI203 overcomes resistance to ABT-199 (venetoclax) by downregulation of BFL-1/A1 in in vitro and in vivo models of MYC+/BCL2+ double hit lymphoma.
ゼブラフィッシュ Tg(6xTcf/LefBS-miniP:d2EGFP) isi04 Bromodomain and Extraterminal (BET) Proteins Regulate Hepatocyte Proliferation in Hepatocyte-Driven Liver Regeneration.
ヒト・動物細胞 StromaNKtert(RCB2350) Pharmacological modulation of CXCR4 cooperates with BET bromodomain inhibition in diffuse large B-cell lymphoma.
ヒト・動物細胞 HCT116(RCB2979) , MKN45(RCB1001) Inhibition of AURKA Reduces Proliferation and Survival of Gastrointestinal Cancer Cells With Activated KRAS by Preventing Activation of RPS6KB1.
ヒト・動物細胞 RBE(RCB1292) Isocitrate dehydrogenase 1 mutation sensitizes intrahepatic cholangiocarcinoma to the BET inhibitor JQ1.
ヒト・動物細胞 TE-1(RCB1894) Targeted inhibition of the COP9 signalosome for treatment of cancer.
ヒト・動物細胞 Lu-165(RCB1184) MYCL is a target of a BET bromodomain inhibitor, JQ1, on growth suppression efficacy in small cell lung cancer cells.
遺伝子材料 CSII-CMV-MCS-IRES2-Venus (RDB04383) The novel orally active proteasome inhibitor K-7174 exerts anti-myeloma activity in vitro and in vivo by down-regulating the expression of class I histone deacetylases.
一般微生物 JCM 6384 Novel semisynthetic antibiotics from caprazamycins A-G: caprazene derivatives and their antibacterial activity.
ヒト・動物細胞 MC3T3-E1(RCB1126) Skeletal protein protection: the mode of action of an anti-osteoporotic marine alkaloid, norzoanthamine.
ヒト・動物細胞 HE19(RCB2239) An analog of BIX-01294 selectively inhibits a family of histone H3 lysine 9 Jumonji demethylases.