RRC ID 44720
著者 Kimura R, Rokkaku T, Takeda S, Senba M, Mori N.
タイトル Cytotoxic effects of fucoidan nanoparticles against osteosarcoma.
ジャーナル Mar Drugs
Abstract In this study, we analyzed the size-dependent bioactivities of fucoidan by comparing the cytotoxic effects of native fucoidan and fucoidan lipid nanoparticles on osteosarcoma in vitro and in vivo. In vitro experiments indicated that nanoparticle fucoidan induced apoptosis of an osteosarcoma cell line more efficiently than native fucoidan. The more potent effects of nanoparticle fucoidan, relative to native fucoidan, were confirmed in vivo using a xenograft osteosarcoma model. Caco-2 cell transport studies showed that permeation of nanoparticle fucoidan was higher than native fucoidan. The higher bioactivity and superior bioavailability of nanoparticle fucoidan could potentially be utilized to develop novel therapies for osteosarcoma.
巻・号 11(11)
ページ 4267-78
公開日 2013-10-30
DOI 10.3390/md11114267
PII md11114267
PMID 24177673
PMC PMC3853727
MeSH Animals Biological Availability Caco-2 Cells Carcinogenesis / drug effects Cell Line, Tumor Female Humans Lung / drug effects Mice Mice, Inbred C3H Nanoparticles / administration & dosage* Osteosarcoma / drug therapy* Permeability Polysaccharides / pharmacology*
IF 4.073
引用数 30
WOS 分野 CHEMISTRY, MEDICINAL
オルトメトリクス指標
オルトメトリクス指標項目
最多言及媒体 Patent(IFI CLAIMS)
各媒体での言及数の合計 2
過去6か月間でのオルトメトリクス指標の変動値 0.0
リソース情報
ヒト・動物細胞 CACO-2(RCB0988)