RRC ID 74368
Author Susumu Shinya, Kentaro Kawai, Naoki Kobayashi, Yukiko Karuo, Atsushi Tarui, Kazuyuki Sato, Masato Otsuka, Masaaki Omote
Title Fluorophenylalkyl-substituted cyanoguanidine derivatives as bacteria-selective MATE transporter inhibitors for the treatment of antibiotic-resistant infections
Journal Bioorganic & Medicinal Chemistry
Volume 74
Pages 117042
Published 2022-11-1
DOI 10.1016/j.bmc.2022.117042
PMID 36215813
MeSH Anti-Bacterial Agents / pharmacology Anti-Infective Agents* / pharmacology Bacteria / metabolism Bacterial Proteins / metabolism Humans Membrane Transport Proteins Norfloxacin* / pharmacology
IF 3.073
Resource
Prokaryotes E. coli