RRC ID 10968
Author Ogawa A, Tomita N, Kikuchi N, Sando S, Aoyama Y.
Title Aptamer selection for the inhibition of cell adhesion with fibronectin as target.
Journal Bioorg Med Chem Lett
Abstract An affinity column immobilizing a decapeptide H(2)N-RGDSPASSKP-CO(2)H was used to select RGD-binding aptamers from a pool of 86-mer single-strand oligodeoxynucleotides (ODNs) containing a random 40-mer sequence. The enriched library thus obtained was further selected against adsorbed fibronectin and individual aptamers were monocloned in E. coli and sequenced to give a couple of highly homologous ODNs, which indeed inhibited fibronectin-integrin mediated cell adhesion.
Volume 14(15)
Pages 4001-4
Published 2004-8-2
DOI 10.1016/j.bmcl.2004.05.042
PII S0960894X04006936
PMID 15225715
MeSH Amino Acid Sequence Animals Base Sequence Cell Adhesion / drug effects* Cell Line Cricetinae Fibronectins / antagonists & inhibitors Fibronectins / physiology* Kidney Models, Molecular Molecular Sequence Data Oligopeptides / chemical synthesis* Oligopeptides / pharmacology* Protein Conformation
IF 2.572
Times Cited 14
WOS Category CHEMISTRY, ORGANIC CHEMISTRY, MEDICINAL
Resource
Human and Animal Cells BHK-21(RCB1423)