RRC ID 73002
Author Eguchi T, Kanai S, Kakinuma K, Okazaki T, Mizoue K.
Title Synthesis of NG-061 and its analogs, and their biological evaluation as an enhancer of nerve growth factor.
Journal Chem Pharm Bull (Tokyo)
Abstract A novel potentiator of nerve growth factor (NGF), NG-061, which had been isolated from the fermentation broth of Penicillium minioluteum F-4627, was synthesized from methoxybenzoquinone and phenylacetylhydrazine in a single step. A series of acyl hydrazone derivatives were also synthesized and their potentiator activity of neurotrophic effect of NGF on neurite outgrowth was evaluated by assay with a rat pheochromocytoma cell line PC12.
Volume 48(10)
Pages 1470-3
Published 2000-10-1
DOI 10.1248/cpb.48.1470
PMID 11045453
MeSH Animals Drug Evaluation, Preclinical Hydrazines / chemical synthesis* Hydrazines / chemistry Hydrazines / pharmacology Molecular Structure Nerve Growth Factor / agonists* PC12 Cells Phenylacetates / chemical synthesis* Phenylacetates / chemistry Phenylacetates / pharmacology Rats Spectrum Analysis
IF 1.416
Resource
Human and Animal Cells PC-12(RCB0009)