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論文 - 一覧

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  • 検索条件 : 絞込み (MeSH = Enzyme Inhibitors / chemistry)
生物種 リソース名 タイトル
一般微生物 JCM 13857 Mass spectrometry-guided discovery of new analogs of bicyclic phosphotriester salinipostin and evaluation of their monoacylglycerol lipase inhibitory activity.
ヒト・動物細胞 HL60(RCB0041) Synthesis of eight stereoisomers of pochonicine: nanomolar inhibition of β-N-acetylhexosaminidases.
原核生物(枯草菌) Armeniaspirols inhibit the AAA+ proteases ClpXP and ClpYQ leading to cell division arrest in Gram-positive bacteria.
ヒト・動物細胞 HCE-T(RCB2280) Identification of sulfonic acids as efficient ecto-5'-nucleotidase inhibitors.
ヒト・動物細胞 K562(RCB0027) Effect of a novel antibiotic, heliquinomycin, on DNA helicase and cell growth.
ヒト・動物細胞 HL-60(RCB3683) Inhibitory Effect of Isoflavones from Erythrina poeppigiana on the Growth of HL-60 Human Leukemia Cells through Inhibition of Glyoxalase I.
ヒト・動物細胞 B16 , SK-MEL-28(RCB1930) WP1066, a small molecule inhibitor of the JAK/STAT3 pathway, inhibits ceramide glucosyltransferase activity.
ヒト・動物細胞 HF19(RCB0210) Synthesis, docking, cytotoxicity, and LTA4H inhibitory activity of new gingerol derivatives as potential colorectal cancer therapy.
ヒト・動物細胞 TGBC11TKB(RCB1148) Human SHMT inhibitors reveal defective glycine import as a targetable metabolic vulnerability of diffuse large B-cell lymphoma.
ヒト・動物細胞 HGC-27(RCB0500) Synthesis and antitumor activity of novel benzimidazole-5-carboxylic acid derivatives and their transition metal complexes as topoisomerease II inhibitors.
ヒト・動物細胞 WI-38(RCB0702) , HeLa Identification of small molecule inhibitors of human COQ7.
ヒト・動物細胞 ST2(RCB0224) FR177995, a novel vacuolar ATPase inhibitor, exerts not only an inhibitory effect on bone destruction but also anti-immunoinflammatory effects in adjuvant-induced arthritic rats.
ヒト・動物細胞 MH7A(RCB1512) Preparative separation of the flavonoid fractions from Periploca forrestii Schltr. ethanol extracts using macroporous resin combined with HPLC analysis and evaluation of their biological activities.
ヒト・動物細胞 HeLa(RCB0007) Identification of Small-Molecule Inhibitors of Human Golgi Mannosidase via a Drug Repositioning Screen.
ヒト・動物細胞 NIH:OVCAR-3(RCB2135) , HeLa(RCB0007) A novel Golgi mannosidase inhibitor: Molecular design, synthesis, enzyme inhibition, and inhibition of spheroid formation.
ヒト・動物細胞 MCF7(RCB1904) Discovery of gamma-mangostin from Garcinia mangostana as a potent and selective natural SIRT2 inhibitor.
ヒト・動物細胞 MCF7(RCB1904) , HeLa , Hep G2 , HCT116(RCB2979) Design, Synthesis and Anticancer Evaluation of New Substituted Thiophene-Quinoline Derivatives.
ヒト・動物細胞 293(RCB1637) Identification of ryuvidine as a KDM5A inhibitor.
遺伝子材料 Histac pcDNA3.1 (RDB12840) Live-cell studies of p300/CBP histone acetyltransferase activity and inhibition.
ショウジョウバエ 4097R–1 , 4097R-2 Proteasome activity determines pupation timing through the degradation speed of timer molecule Blimp-1.