Reference - Detail
RRC ID | 68588 |
---|---|
Author | Koga K, Yoshinaga M, Uematsu Y, Nagai Y, Miyakoshi N, Shimoda Y, Fujinaga M, Minamimoto T, Zhang MR, Higuchi M, Ohtake N, Suhara T, Chaki S. |
Title | TASP0434299: A Novel Pyridopyrimidin-4-One Derivative as a Radioligand for Vasopressin V1B Receptor. |
Journal | J Pharmacol Exp Ther |
Volume | 357(3) |
Pages | 495-508 |
Published | 2016-6-1 |
DOI | 10.1124/jpet.116.232942 |
PII | jpet.116.232942 |
PMID | 27029585 |
MeSH | Animals Binding, Competitive Biological Transport Carbon Radioisotopes HEK293 Cells Humans Macaca mulatta Male Pituitary Gland / metabolism Positron-Emission Tomography Protein Binding Pyridines / metabolism* Pyrimidines / metabolism* Pyrimidinones / metabolism* Radioactive Tracers Radioligand Assay Rats Rats, Sprague-Dawley Receptors, Vasopressin / metabolism* |
IF | 3.561 |
Resource | |
Human and Animal Cells | LLC-GA5-CoL300(RCB0872) |