RRC ID 68588
Author Koga K, Yoshinaga M, Uematsu Y, Nagai Y, Miyakoshi N, Shimoda Y, Fujinaga M, Minamimoto T, Zhang MR, Higuchi M, Ohtake N, Suhara T, Chaki S.
Title TASP0434299: A Novel Pyridopyrimidin-4-One Derivative as a Radioligand for Vasopressin V1B Receptor.
Journal J Pharmacol Exp Ther
Volume 357(3)
Pages 495-508
Published 2016-6-1
DOI 10.1124/jpet.116.232942
PII jpet.116.232942
PMID 27029585
MeSH Animals Binding, Competitive Biological Transport Carbon Radioisotopes HEK293 Cells Humans Macaca mulatta Male Pituitary Gland / metabolism Positron-Emission Tomography Protein Binding Pyridines / metabolism* Pyrimidines / metabolism* Pyrimidinones / metabolism* Radioactive Tracers Radioligand Assay Rats Rats, Sprague-Dawley Receptors, Vasopressin / metabolism*
IF 3.561
Resource
Human and Animal Cells LLC-GA5-CoL300(RCB0872)