Reference - Detail
| RRC ID | 68588 |
|---|---|
| Author | Koga K, Yoshinaga M, Uematsu Y, Nagai Y, Miyakoshi N, Shimoda Y, Fujinaga M, Minamimoto T, Zhang MR, Higuchi M, Ohtake N, Suhara T, Chaki S. |
| Title | TASP0434299: A Novel Pyridopyrimidin-4-One Derivative as a Radioligand for Vasopressin V1B Receptor. |
| Journal | J Pharmacol Exp Ther |
| Volume | 357(3) |
| Pages | 495-508 |
| Published | 2016-6-1 |
| DOI | 10.1124/jpet.116.232942 |
| PII | jpet.116.232942 |
| PMID | 27029585 |
| MeSH | Animals Binding, Competitive Biological Transport Carbon Radioisotopes HEK293 Cells Humans Macaca mulatta Male Pituitary Gland / metabolism Positron-Emission Tomography Protein Binding Pyridines / metabolism* Pyrimidines / metabolism* Pyrimidinones / metabolism* Radioactive Tracers Radioligand Assay Rats Rats, Sprague-Dawley Receptors, Vasopressin / metabolism* |
| IF | 3.561 |
| Resource | |
| Human and Animal Cells | LLC-GA5-CoL300(RCB0872) |