RRC ID 68588
著者 Koga K, Yoshinaga M, Uematsu Y, Nagai Y, Miyakoshi N, Shimoda Y, Fujinaga M, Minamimoto T, Zhang MR, Higuchi M, Ohtake N, Suhara T, Chaki S.
タイトル TASP0434299: A Novel Pyridopyrimidin-4-One Derivative as a Radioligand for Vasopressin V1B Receptor.
ジャーナル J Pharmacol Exp Ther
巻・号 357(3)
ページ 495-508
公開日 2016-6-1
DOI 10.1124/jpet.116.232942
PII jpet.116.232942
PMID 27029585
MeSH Animals Binding, Competitive Biological Transport Carbon Radioisotopes HEK293 Cells Humans Macaca mulatta Male Pituitary Gland / metabolism Positron-Emission Tomography Protein Binding Pyridines / metabolism* Pyrimidines / metabolism* Pyrimidinones / metabolism* Radioactive Tracers Radioligand Assay Rats Rats, Sprague-Dawley Receptors, Vasopressin / metabolism*
IF 3.561
リソース情報
ヒト・動物細胞 LLC-GA5-CoL300(RCB0872)