RRC ID 61368
Author Lianbao Ye, Yuanxin Tian, Zhonghuang Li, Hong Jin, Zhengguang Zhu, Shanhe Wan, Junyan Zhang, Pengjiu Yu, Jiajie Zhang, Shuguang Wu
Title Design, synthesis and molecular docking studies of some novel spiro[indoline-3, 4′-piperidine]-2-ones as potential c-Met inhibitors
Journal European Journal of Medicinal Chemistry
Volume 50
Pages 370-375
Published 2012-4-1
DOI 10.1016/j.ejmech.2012.02.016
PMID 22381355
MeSH Binding Sites Blotting, Western Cell Proliferation / drug effects Drug Design* Drug Discovery Fluorescence Resonance Energy Transfer Humans Inhibitory Concentration 50 Models, Molecular Molecular Structure Piperidines / chemistry* Protein Kinase Inhibitors / chemical synthesis* Protein Kinase Inhibitors / pharmacology* Proto-Oncogene Proteins c-met / antagonists & inhibitors* Stomach Neoplasms / drug therapy* Stomach Neoplasms / metabolism Structure-Activity Relationship Tumor Cells, Cultured
IF 5.573
Resource
Human and Animal Cells MKN45(RCB1001)