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論文 - 詳細
RRC ID
65063
著者
Kikuchi A, Suzuki T, Nakazawa T, Iizuka M, Nakayama A, Ozawa T, Kameda M, Shindoh N, Terasaka T, Hirano M, Kuromitsu S.
タイトル
ASP5878, a selective FGFR inhibitor, to treat FGFR3-dependent urothelial cancer with or without chemoresistance.
ジャーナル
Cancer Sci
巻・号
108(2)
ページ
236-242
公開日
2017-2-1
DOI
10.1111/cas.13124
PMID
27885740
PMC
PMC5329164
MeSH
ATP Binding Cassette Transporter, Subfamily B / metabolism
Antineoplastic Agents / pharmacology
Body Weight / drug effects
Cell Line, Tumor
Cell Proliferation / drug effects
DNA-Binding Proteins / metabolism
Deoxycytidine / analogs & derivatives
Deoxycytidine / pharmacology
Doxorubicin / pharmacology
Drug Resistance, Neoplasm / drug effects
Drug Resistance, Neoplasm / genetics
Gemcitabine
Gene Fusion
Humans
Molecular Targeted Therapy*
Point Mutation
Pyrazoles / pharmacology*
Pyrimidines / pharmacology*
Receptor, Fibroblast Growth Factor, Type 3 / antagonists & inhibitors
Receptor, Fibroblast Growth Factor, Type 3 / genetics*
Transcription Factors / metabolism
Urologic Neoplasms / drug therapy*
Urologic Neoplasms / genetics
Urologic Neoplasms / metabolism
IF
4.966
リソース情報
ヒト・動物細胞
BOY-12E(RCB2627)
JMSU1(RCB2227)